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Q Filgotinib用途是什么?

Question time:6/10/2021 11:18:41 AM

Describe:Filgotinib是做什么用的?哪里可以用到Filgotinib?

A
admin 2021-06-30 13:02
Filgotinib一种高效、选择性的JAK1抑制剂,能够有效抑制JAK1、JAK2、JAK3和TYK2的活性,IC50值分别为10nM、28nM、810nM和116nM。Filgotinib is a potent and selective JAK1 inhibitor. It is considered a promising agent as it inhibits JAK1 selectively. Filgotinib displayed a selectivity of 30-fold fo

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