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Q P276-00用途是什么?

Question time:8/30/2021 9:30:19 AM

Describe:P276-00是做什么用的?哪里可以用到P276-00?

A
admin 2021-09-09 14:28
P276-00Riviciclib盐酸盐用途Riviciclib hydrochloride (P276-00) 是有效的 CDK 抑制剂,抑制 CDK9-cyclinT1,CDK4-cyclin D1,CDK1-cyclinB,CDK2-cyclin A,CDK2-cyclin E,CDK6-cyclin D3,CDK9-cyclin H 的IC50分别为 20 nM, 63 nM,79 nM,224 nM,2500 nM,396 nM,2900 nM。Riviciclib hydrochloride 对 Cisplatin 耐药性细胞具有抗肿瘤活性。

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